| Title | Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors |
| Publication Type | Journal Article |
| Year of Publication | 2018 |
| Authors | Shadrick WR, Slavish PJ, Chai SC, Waddell B, Connelly M, Low JA, Tallant C, Young BM, Bharatham N, Knapp S, Boyd VA, Morfouace M, Roussel MF, Chen T, Lee RE, R. Guy K, Shelat AA, Potter PM |
| Journal | Bioorganic & Medicinal Chemistry |
| Volume | 26 |
| Pagination | 25 - 36 |
| ISSN | 0968-0896 |
| URL | http://www.sciencedirect.com/science/article/pii/S0968089617315948 |
| DOI | 10.1016/j.bmc.2017.10.042 |
